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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 2' and Ligand = 'BDBM50028125'
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
GlaxoSmithKline R&D
Curated by
ChEMBL
Ligand
BDBM50028125
(CHEMBL3353990)
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Affinity Data
IC50: 794nM
Assay Description:
Displacement of biotinylated tetra-acetylated histone H4 from His6-tagged BRD2 (1 to 473 aa) (unknown origin) after 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q23R0VGR
PubMed