Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3' and Ligand = 'BDBM50443232'
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50443232(CHEMBL3086883)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of human 6x-His-tagged BRD3 bromodomain 1 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3PRQPubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50443232(CHEMBL3086883)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of fluorescein-labeled MS574 from recombinant human BRD3 BrD1 after 1 hr by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1NCFPubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50443232(CHEMBL3086883)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Inhibition of human 6x-His-tagged BRD3 bromodomain 2 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3PRQPubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50443232(CHEMBL3086883)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Displacement of fluorescein-labeled MS574 from recombinant human BRD3 BrD2 after 1 hr by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZW1NCFPubMed