Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM223494'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
DANA-FARBER CANCER INSTITUTE, INC.

US Patent
LigandPNGBDBM223494(US10407441, Compound JQ33 | US9320741, JQ33)copy SMILEScopy InChI
Affinity DataIC50: 29.5nMpH: 7.4 T: 2°CAssay Description:BRD4(2): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KP811PUS Patent
TargetBromodomain-containing protein 4(Homo sapiens (Human))
DANA-FARBER CANCER INSTITUTE, INC.

US Patent
LigandPNGBDBM223494(US10407441, Compound JQ33 | US9320741, JQ33)copy SMILEScopy InChI
Affinity DataIC50: 85nMpH: 7.4 T: 2°CAssay Description:BRD4(1): Assays were performed as described previously with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KP811PUS Patent