Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50183564'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 5.86E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG

Curated by ChEMBL
LigandPNGBDBM50183564(CHEMBL3822990)copy SMILEScopy InChI
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD2 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1MJZPubMed