Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50504153'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cellzome

Curated by ChEMBL
LigandPNGBDBM50504153(CHEMBL4568748)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from His6-tagged BRD4 BD2 (1 to 477 residues)/BD1 Y97A mutant (unknown origin) after 30 mins by TR-FR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3VZVPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cellzome

Curated by ChEMBL
LigandPNGBDBM50504153(CHEMBL4568748)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+4nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant (unknown origin) after 30 mins by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3VZVPubMed