Found 1 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50539794'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Illinois at Chicago
Curated by ChEMBL
University of Illinois at Chicago
Curated by ChEMBL
Affinity DataIC50: 175nMAssay Description:Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubat...More data for this Ligand-Target Pair