Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50544616'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
GSK

Curated by ChEMBL
LigandPNGBDBM50544616(CHEMBL4635329)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of Alexa Fluor 647 labelled I-BET762 from N-terminal His6-tagged human BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant expressed in Escher...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348Q0NPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
GSK

Curated by ChEMBL
LigandPNGBDBM50544616(CHEMBL4635329)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of Alexa Fluor 647 labelled I-BET762 from N-terminal His6-tagged human BRD4 BD2 (1 to 477 residues)/BD1 Y97A mutant expressed in Escheri...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348Q0NPubMed