Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
Found
2
Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [44-168]' and Ligand = 'BDBM205438'
Target
Bromodomain-containing protein 4 [44-168]
(Homo sapiens (Human))
Dana-Farber Cancer Institute
Ligand
BDBM205438
(6S+IBET-PEG2 (19))
copy SMILES
copy InChI
Affinity Data
IC50: 58.6nM
pH: 7.5 T: 2°C
Assay Description:
Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2VQ31HW
PubMed
Target
Bromodomain-containing protein 4 [44-168]
(Homo sapiens (Human))
Dana-Farber Cancer Institute
Ligand
BDBM205438
(6S+IBET-PEG2 (19))
copy SMILES
copy InChI
Affinity Data
Kd: 0.0620nM
Assay Description:
Refer to DiscoverX
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2VQ31HW
PubMed