Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [49-170]/DNA damage-binding protein 1/Protein cereblon' and Ligand = 'BDBM511636'
LigandPNGBDBM511636(US11059801, Compound dBET45)copy SMILES
Affinity DataIC50: 1.54E+4nMAssay Description:AlphaScreen technology was used to detect CRBN-DDB1/BRD4 dimerization induced by dBET molecules. In brief, GST-BRD4[49-170] (Sigma Aldrich) and CRBN-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2G44TFMUS Patent