Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [75-147]' and Ligand = 'BDBM249294'
TargetBromodomain-containing protein 4 [75-147](Homo sapiens (Human))
Gilead Sciences, Inc.

US Patent
LigandPNGBDBM249294(US10017501, Compound 1020-90 | US9458145, 1020-90)copy SMILEScopy InChI
Affinity DataIC50: 29.9nMpH: 7.5 T: 2°CAssay Description:Binding of the bromodomain BRD4-I to an acetylated histone H4 peptide was measured using a bead-based Amplified Luminescent Proximity Homogeneous Ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1W53US Patent
TargetBromodomain-containing protein 4 [75-147](Homo sapiens (Human))
Gilead Sciences, Inc.

US Patent
LigandPNGBDBM249294(US10017501, Compound 1020-90 | US9458145, 1020-90)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Binding of the two tandem bromodomains, BRD4-1 and BRD4-2, to an acetylated histone H4 peptide was measured using a homogeneous time resolved fluores...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4M3ZUS Patent
TargetBromodomain-containing protein 4 [75-147](Homo sapiens (Human))
Gilead Sciences, Inc.

US Patent
LigandPNGBDBM249294(US10017501, Compound 1020-90 | US9458145, 1020-90)copy SMILEScopy InChI
Affinity DataIC50: 110nMpH: 7.5 T: 2°CAssay Description:Binding of the two tandem bromodomains, BRD4-1 and BRD4-2, to an acetylated histone H4 peptide was measured using a homogeneous time resolved fluores...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1W53US Patent