Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 3' and Ligand = 'BDBM50159702'
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50159702(CHEMBL3786670)copy SMILEScopy InChI
Affinity DataEC50:  759nMAssay Description:Positive allosteric modulation of ProLink2-tagged wild type CXCR3 (unknown origin) expressed in HEK293T cells assessed as beta-arrestin-2 recruitment...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72KBRPubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50159702(CHEMBL3786670)copy SMILEScopy InChI
Affinity DataEC50:  1.15E+3nMAssay Description:Positive allosteric modulation of human CXCR3 expressed in HEK293T cell membranes after 30 mins by [35S]GTPgammaS incorporation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72KBRPubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Friedrich Alexander University

Curated by ChEMBL
LigandPNGBDBM50159702(CHEMBL3786670)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Positive allosteric modulation of ProLink1-tagged wild type CXCR3 (unknown origin) expressed in HEK293T cells assessed as beta-arrestin-2 recruitment...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72KBRPubMed