Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 6' and Ligand = 'BDBM50539470'
TargetC-X-C chemokine receptor type 6(Homo sapiens)
Sanford Burnham Prebys Medical Discovery Institute

Curated by ChEMBL
LigandPNGBDBM50539470(CHEMBL4642230)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077T6PubMed
TargetC-X-C chemokine receptor type 6(Homo sapiens)
Sanford Burnham Prebys Medical Discovery Institute

Curated by ChEMBL
LigandPNGBDBM50539470(CHEMBL4642230)copy SMILEScopy InChI
Affinity DataIC50: 7.90E+3nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077T6PubMed