Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'CDK-activating kinase assembly factor MAT1' and Ligand = 'BDBM59227'
TargetCDK-activating kinase assembly factor MAT1(Homo sapiens (Human))
GPC Biotech, Inc.

LigandPNGBDBM59227(Pyrazolopyrimidone analog, RGB-286147)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of in vitro kinase activity of purified CDKs.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3BR6PubMed