Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'CREB-binding protein' and Ligand = 'BDBM50370181'
TargetCREB-binding protein(Homo sapiens (Human))TBA
LigandPNGBDBM50370181(CHEMBL4159382 | US11117865, Compound ZL0454)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetCREB-binding protein(Homo sapiens (Human))TBA
LigandPNGBDBM50370181(CHEMBL4159382 | US11117865, Compound ZL0454)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CBP (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X069KMPubMed