Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Calcitonin gene-related peptide type 1 receptor' and Ligand = 'BDBM50192538'
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50192538((R)-N-(2-oxo-5-phenyl-1-(2,2,2-trifluoroethyl)-2,3...)copy SMILEScopy InChI
Affinity DataKi:  51nMAssay Description:Displacement of [125I]CGRP from human recombinant CGRP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QNXPubMed
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50192538((R)-N-(2-oxo-5-phenyl-1-(2,2,2-trifluoroethyl)-2,3...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Activity at CGRP receptor assessed as inhibition of CGRP-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QNXPubMed