Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Calmodulin-domain protein kinase 1' and Ligand = 'BDBM50148727'
TargetCalmodulin-domain protein kinase 1(Toxoplasma gondii)
University of Washington Through its Center For Commercialization

US Patent
LigandPNGBDBM50148727(CHEMBL3770430 | US9518026, Example 64 | US9956214,...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BV7JN4US Patent
TargetCalmodulin-domain protein kinase 1(Toxoplasma gondii)
University of Washington Through its Center For Commercialization

US Patent
LigandPNGBDBM50148727(CHEMBL3770430 | US9518026, Example 64 | US9956214,...)copy SMILEScopy InChI
Affinity DataIC50: 115nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23J3G91US Patent
TargetCalmodulin-domain protein kinase 1(Toxoplasma gondii)
University of Washington Through its Center For Commercialization

US Patent
LigandPNGBDBM50148727(CHEMBL3770430 | US9518026, Example 64 | US9956214,...)copy SMILEScopy InChI
Affinity DataIC50: 115nMAssay Description:Inhibition of Toxoplasma gondii CDPK1 assessed as ATP consumption using (Biotin-C6-PLARTLSVAGLPGKK) as substrate after 90 mins by luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3GXDPubMed