Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50279126'
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279126(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-m...)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50279126(2-[5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-m...)copy SMILEScopy InChI
Affinity DataEC50:  8.5nMAssay Description:Inverse agonist activity at human recombinant CB1R expressed in HEK293 cells assessed as inhibition of CP55940-stimulated Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W99Z4PubMed