Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50239215'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor Corporation

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP55940 from human cloned CB2 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G73DK3PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor Corporation

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP 55940 from human CB2 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9QCJPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor Corporation

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2701MPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor Corporation

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)copy SMILEScopy InChI
Affinity DataEC50:  21nMAssay Description:Agonist activity at human cloned CB2 receptor by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P2701MPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor Corporation

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)copy SMILEScopy InChI
Affinity DataEC50:  21nMAssay Description:Agonist activity at human cloned CB2 receptor assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G73DK3PubMed