Compile Data Set for Download or QSAR
Found 10 Enz. Inhib. hit(s) with Target = 'Casein kinase II subunit alpha 3' and Ligand = 'BDBM50530315'
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as reduction in STAT3 phosphorylation at Y705 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in p21 phosphorylation at Thr145 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  3.20E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in Akt1 phosphorylation at Ser129 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in alpha-catenin phosphorylation at Ser641 assuming basal level of non-responsive P-alpha...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in p21 phosphorylation at Thr145 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as reduction in STAT3 phosphorylation at Y705 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  9.00E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in alpha-catenin phosphorylation at Ser641 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  9.00E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in alpha-catenin phosphorylation at Ser641 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  3.20E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in Akt1 phosphorylation at Ser129 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Universit£ de Lyon

Curated by ChEMBL
LigandPNGBDBM50530315(CHEMBL4520531)copy SMILEScopy InChI
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of CK2 in human 786-0 cells assessed as decrease in alpha-catenin phosphorylation at Ser641 assuming basal level of non-responsive P-alpha...More data for this Ligand-Target Pair