Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50008170'
TargetCholecystokinin receptor type A(RAT)
Universitá di Siena

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataKi:  129nMAssay Description:Binding affinity against Cholecystokinin type A receptor using [125I]-(BH)-CCK-8 as radioligand in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222SVDPubMed
TargetCholecystokinin receptor type A(RAT)
Universitá di Siena

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of binding of [125I]- CCK-33 to rat pancreasMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29K4BTPPubMed
TargetCholecystokinin receptor type A(RAT)
Universitá di Siena

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]-CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6J92
TargetCholecystokinin receptor type A(RAT)
Universitá di Siena

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5W11PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008170(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of binding of [125I]- CCK-33 to guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29K4BTPPubMed