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Affinity DataKi: 129nMAssay Description:Binding affinity against Cholecystokinin type A receptor using [125I]-(BH)-CCK-8 as radioligand in rat pancreas.More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of binding of [125I]- CCK-33 to rat pancreasMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]-CCK-OP radioligand from Cholecystokinin type A receptor in rat pancreatic acinar membrane binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Concentration required to inhibit by 50% specific binding of [125I](BH)-CCK-8 to cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(Cavia porcellus)
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp& Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of binding of [125I]- CCK-33 to guinea pig cortexMore data for this Ligand-Target Pair
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