Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Corticotropin-releasing factor receptor 1' and Ligand = 'BDBM50398578'
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50398578(CHEMBL2179183 | US8530504, 27)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Displacement of [125I]CRF from human CRF1 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD202PPubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50398578(CHEMBL2179183 | US8530504, 27)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:A binding competition experiment with CRF was conducted by the SPA (GE Healthcare) method using a 96-well plate.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29885NSUS Patent