Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Cyclin-G-associated kinase' and Ligand = 'BDBM50537135'
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50537135(CHEMBL4592501)copy SMILEScopy InChI
Affinity DataKd:  48nMAssay Description:Binding affinity to human wild type partial length GAK (G13 to Y338 residues) expressed in bacterial expression system by KinomeScan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9FC5PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50537135(CHEMBL4592501)copy SMILEScopy InChI
Affinity DataKd:  21nMAssay Description:Binding affinity to biotinylated human GAK (13 to 338 residues) expressed in Escherichia coli incubated for 1.5 hrs by fluorescent tracer dependent T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed