Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 1' and Ligand = 'BDBM50232241'
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50232241(4-(2-Chlorophenyl)-9-hydroxy-6-(3-hydroxypropyl)-p...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human Cdc2 kinase PY15 phosphorylation in HT29 cells by Western blotMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2XC3PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50232241(4-(2-Chlorophenyl)-9-hydroxy-6-(3-hydroxypropyl)-p...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of Cdc2 Tyr15 phosphorylation in human HT29 cells by western blotMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36MCPubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50232241(4-(2-Chlorophenyl)-9-hydroxy-6-(3-hydroxypropyl)-p...)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:Inhibition of Cdc2/cyclin B assessed as inhibition of histone H1 phosphorylation in human HT29 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36MCPubMed