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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 2/G1/S-specific cyclin-E1' and Ligand = 'BDBM7667'
Target
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1
(Homo sapiens (Human))
AstraZeneca
Ligand
BDBM7667
(4-[(4-{6-bromoimidazo[1,2-a]pyridin-3-yl}pyrimidin...)
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Affinity Data
IC50: 3nM
pH: 7.0 T: 2°C
Assay Description:
The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2XG9PCF
PubMed