Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 3/G1/S-specific cyclin-E1' and Ligand = 'BDBM50113281'
TargetCyclin-dependent kinase 3/G1/S-specific cyclin-E1(Homo sapiens (Human))
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM50113281(AT-7519)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged CDK3/full-length human N-terminal GST-tagged Cyclin E expressed in baculovirus inf...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q21J2PubMed
TargetCyclin-dependent kinase 3/G1/S-specific cyclin-E1(Homo sapiens (Human))
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM50113281(AT-7519)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of CDK3/cyclin E (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K3WPubMed
TargetCyclin-dependent kinase 3/G1/S-specific cyclin-E1(Homo sapiens (Human))
University of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM50113281(AT-7519)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of CDK3/cyclin E1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K3WPubMed