Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 5 activator 1' and Ligand = 'BDBM50215927'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Macquarie University

Curated by ChEMBL
LigandPNGBDBM50215927(4-(1H-pyrrol-2-yl)-1H-imidazo[4,5-c]pyridin-2-amin...)copy SMILEScopy InChI
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma-32P] ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3NMTPubMed