Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 5 activator 1' and Ligand = 'BDBM7266'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£t Braunschweig

Curated by ChEMBL
LigandPNGBDBM7266(14-bromo-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)copy SMILEScopy InChI
Affinity DataIC50: 850nMAssay Description:Inhibition of recombinant CDK5/p25 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2X22PubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£t Braunschweig

Curated by ChEMBL
LigandPNGBDBM7266(14-bromo-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)copy SMILEScopy InChI
Affinity DataIC50: 850nMAssay Description:Inhibition of Cyclin-dependent kinase 5 (CDK5)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X067TXPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Technische Universit£t Braunschweig

Curated by ChEMBL
LigandPNGBDBM7266(14-bromo-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 assessed as incorporation of [gamma-33P]-ATP into histone H1 substrate after 30 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21836T2PubMed