Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 5 activator 1' and Ligand = 'BDBM7401'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
C.N.R.S.

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0N3ZPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
C.N.R.S.

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:inhibition of human recombinant CDK5/p25 using histone H1 as substrate by scintillation counting in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VHKPubMed