Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 5 activator 1' and Ligand = 'BDBM7534'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
India; Academy of Scientific and Innovative Research (AcSIR)

Curated by ChEMBL
LigandPNGBDBM7534(1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK5/p25 (unknown origin) expressed in Escherichia coli using histone as substrate in presence of [gamma32P]ATP after 10 mins by scinti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WQ074MPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
India; Academy of Scientific and Innovative Research (AcSIR)

Curated by ChEMBL
LigandPNGBDBM7534(1H-pyrazolo[3,4-b]quinoxalin-3-amine | pyrazolo[3,...)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of GST-tagged CDK5/p25 (unknown origin) expressed in Baculovirus infected Sf9 cells using histone H1 as substrate as substrate in presence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB5665PubMed