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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Cytochrome P450 3A4' and Ligand = 'BDBM50265951'
Target
Cytochrome P450 3A4
(Homo sapiens (Human))
University of Washington at Seattle
Ligand
BDBM50265951
(CHEMBL1657 | TAZAROTENE | US9963439, Tazarotene | ...)
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Affinity Data
IC50: 3.15E+3nM
Assay Description:
Compounds were assessed for inhibition (IC50, n=2) of CYP2C8, CYP2C9 and CYP3A4 in pooled human liver microsomes using selective probe substrates at ...
More data for this Ligand-Target Pair
Target Info
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MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
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Ligand Info
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Details
BindingDB Entry DOI:
10.7270/Q2FN18J2
US Patent