Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'D(1A) dopamine receptor' and Ligand = 'BDBM81986'
TargetD(1A) dopamine receptor(Mus musculus (Mouse))
NOVO Industri A/S

Curated by PDSP Ki Database
LigandPNGBDBM81986(3-Methyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]az...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6P1HPubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM81986(3-Methyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]az...)copy SMILEScopy InChI
Affinity DataKi:  8.80nMAssay Description:The compound was evaluated for the dissociation constant for inhibiting the binding of [3H]-SCH- 23390 at dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26H4J17PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM81986(3-Methyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]az...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human dopamine D1 receptor expressed in CHOK1 cells assessed as assessed as increase in beta-arrestin-2 recruitment after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76GX7PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM81986(3-Methyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]az...)copy SMILEScopy InChI
Affinity DataEC50:  0.450nMAssay Description:Agonist activity at human dopamine D1 receptor expressed in CHOK1 cells assessed as reversal of Ro 20-1724 mediated decrease in cAMP accumulation aft...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76GX7PubMed