Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM423299'
TargetD(2) dopamine receptor(Homo sapiens (Human))
NHWA PHARMA. CORPORATION

US Patent
LigandPNGBDBM423299(US10501452, Compound 5)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:D2:Procedures(1) The prepared membrane was applied with appropriate amount of buffer, and homogenizer was used for evenly dispersing. 15 tubes were m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BK1FR6US Patent
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM423299(US10501452, Compound 5)copy SMILEScopy InChI
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]spiperone from D2 receptor in rat striatum measured after 15 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8K6MPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
NHWA PHARMA. CORPORATION

US Patent
LigandPNGBDBM423299(US10501452, Compound 5)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human D2 receptor expressed in CHO-K1 cells assessed as inhibition of dopamine-induced calcium flux incubated for 60 mins at 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8K6MPubMed