Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50164880'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50164880(CHEMBL3800165)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]7-OH-DPAT from human D2 receptor transfected in HEK293 cells measured after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2708393PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50164880(CHEMBL3800165)copy SMILEScopy InChI
Affinity DataKi:  868nMAssay Description:Displacement of [3H]N-methylspiperone from human D2 receptor transfected in HEK293 cells measured after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2708393PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50164880(CHEMBL3800165)copy SMILEScopy InChI
Affinity DataEC50:  68nMAssay Description:Agonist activity at human D2 receptor transfected in HEK293T cells by BRET based G0 activation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2708393PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50164880(CHEMBL3800165)copy SMILEScopy InChI
Affinity DataEC50:  13nMAssay Description:Agonist activity at recombinant human D2 receptor expressing in CHOp cells assessed as receptor mediated stimulation of mitogenesis measured as [3H]t...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2708393PubMed