Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50568760'
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50568760(CHEMBL4846380)copy SMILES
Affinity DataKi:  17nMAssay Description:Displacement of [3H]N-methylspiperone from human D3 receptor expressed in HEK293T cells co-expressing CRE-Luc incubated for 60 mins by microbeta scin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF0245PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50568760(CHEMBL4846380)copy SMILES
Affinity DataEC50:  102nMAssay Description:Agonist activity at human histamine D3 receptor receptor expressed in HEK293T cells co-expressing ELucC by beta arrestin2 recruitment assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF0245PubMed