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TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
WuXi Apptec (Tianjin) Co. Ltd.
Curated by ChEMBL
WuXi Apptec (Tianjin) Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human DNMT1 using polydeoxyinosine polydeoxycytosine DNA as substrate after 15 mins in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
WuXi Apptec (Tianjin) Co. Ltd.
Curated by ChEMBL
WuXi Apptec (Tianjin) Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human DNMT1 enzyme using polydeoxy-inosine polydeoxy-cytosine DNA as substrate incubated for 15 mins in presence of SAM by TR-FRET assa...More data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
WuXi Apptec (Tianjin) Co. Ltd.
Curated by ChEMBL
WuXi Apptec (Tianjin) Co. Ltd.
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of DNMT1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
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