Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'DNA-dependent protein kinase catalytic subunit' and Ligand = 'BDBM50197062'
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Curtin University

Curated by ChEMBL
LigandPNGBDBM50197062(Pilaralisib | SAR-245408 | XL-147)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human DNA-PK by by luciferase-luciferin-coupled chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1TPXPubMed