Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM214798'
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM214798(Dynorphin A (1-17) | YGGFLRRIRPKLK)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM214798(Dynorphin A (1-17) | YGGFLRRIRPKLK)copy SMILEScopy InChI
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]deltorphin-II from human DOR expressed in CHO cell membranes incubated for 2 hrs by liquid scintillation counting based radioliga...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6WWTPubMed
TargetDelta-type opioid receptor(MOUSE)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM214798(Dynorphin A (1-17) | YGGFLRRIRPKLK)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed