Compile Data Set for Download or QSAR
Found 8 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM224024'
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataKi:  14.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23J3BH2PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J965CZPubMed
TargetDelta-type opioid receptor(GUINEA PIG)
SRI International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataKi:  16.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23J3BH2PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Binding affinity to Opioid receptor delta 1 by competitive inhibition of radioligand [3H]-DPDPE using cloned receptors transiently expressed on CHO c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2N3HPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [3H]-DPDPE binding to delta opioid receptor of guinea pig brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936K7PubMed
TargetDelta-type opioid receptor(MOUSE)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Inhibition of delta-selective antagonist binding to opioid receptor of mouse vas dferensMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K936K7PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as calcium mobilization by Fluo-4 AM based fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22809FJPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by PDSP Ki Database
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321H7PubMed