Found 40 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM82551' TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Antagonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of compound 14-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor expressed in HEK293 cells by visible spectrophotometryMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Compound was evaluated for functional opioid activity by stimulation of [35S]GTP-gamma-S, in cloned human Opioid receptor delta 1 transfected into C...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cell membranes after 60 mins by scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of [3H]- diprenorphine from delta-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Compound was evaluated for its binding affinity to CHO cells expressing cloned human Opioid receptor delta 1 by displacement of [3H]Cl-DPDPEMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Binding affinity against cloned human Opioid receptor delta 1 transfected into chinese hamster ovary cells using [3H]Cl-DPDPE as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Ability to displace [3H]DPDPE from human recombinant Opioid receptor delta 1 in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Binding affinity towards human cloned Opioid receptor delta 1 using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Inhibition of [3H]C1-DPDPE binding to human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]C1-DPDPE from human recombinant Opioid receptor delta 1 on CHO cell membranes.More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Inhibition of [3H]diprenorphine binding to rat Opioid receptor delta 1 expressed in C6 cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 6.60nMAssay Description:Displacement of [3H]diprenorphine from human opioid delta receptor expressed in HEK293 cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Antagonist activity on agonist stimulated [35S]GTP-gamma-S, binding in guinea pig caudate membranes (10 uM SNC-80 as the agonist ligand for delta-rec...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of [35S]GTP-gamma-S, binding from Opioid receptor delta 1 in Guinea pig Caudate stimulated by SNC80More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of stimulation of [35S]GTP-gamma-S, binding produced by the selective agonist (SNC-80, delta-receptor), in guinea pig caudate membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Antagonist activity on agonist (SNC-80) stimulated [35S]GTP-gamma-S, binding in cloned delta opioid receptorsMore data for this Ligand-Target Pair
Affinity DataKi: 17.7nMAssay Description:Binding affinity was measured on delta opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity towards cloned human Opioid receptor delta 1 in CHO cell membranes.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:In vitro binding affinity to human Opioid receptor delta 1 on CHO cell membranes using [3H]diprenorphine displacement.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]Naltrindole form human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Binding affinity against Opioid receptor delta 1 was measured in the guinea pig brain membranes using [3H]DADLE in the presence of 1 uM unlabeled DAM...More data for this Ligand-Target Pair
Affinity DataKi: 41.5nMAssay Description:Displacement of [3H]- diprenorphine from mu-K303E-receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Binding affinity for delta opioid receptor was determined using radioligand [3H]DPDPE in Guinea pig brain membranes.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Binding affinity determined on Opioid receptor delta 1 in Guinea pig brain membranes using radioligand [3H]DADLEMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibition of [3H]-DADLE binding to Opioid receptor delta 1 of rat brain tissueMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Binding affinity of compound for opioid receptor delta 1 was determined using [3H]DADLE as radioligand from rat brain tissueMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Binding affinity to delta-opioid receptor of rat brain using [3H]DADLE as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against delta-opioid receptor in mouse vas deferens preparation using DADLEMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Opioid receptor delta 1 by displacing 1 nM [3H]DPDPE in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human delta opioid receptor expressed in HEK cells assessed as inhibition of SNC-80-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human delta opioid receptor assessed as inhibition of SNC80-stimulated [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataEC50: 4.40nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding at human recombinant Opioid receptor delta 1 transfected into CHO cells.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Human BioMolecular Research Institute
Curated by ChEMBL
Human BioMolecular Research Institute
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Agonist activity at human recombinant delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
