Compile Data Set for Download or QSAR
Found 8 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 1' and Ligand = 'BDBM385066'
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F76HN2
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FB56W4
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMAssay Description:The activity of DPP1 was determined by measuring the enzymatic release of aminomethyl coumarin (AMC) from the peptide substrate (H-Gly-Arg-AMC), whic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RJ4MTPUS Patent
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6X5T
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMAssay Description:Examples 1-35: The activity of DPP1 was determined by measuring the enzymatic release of aminomethyl coumarin (AMC) from the peptide substrate (H-Gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q243DZUS Patent
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24X5CXQ
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H99949
TargetDipeptidyl peptidase 1(Homo sapiens (Human))TBA
LigandPNGBDBM385066((2S)-N-{(1S)-2-[4-(7-Chloro-3-methyl-2-oxo-2,3-dih...)copy SMILEScopy InChI
Affinity DataIC50: 13.5nMAssay Description:The activity of DPP1 was determined by measuring the enzymatic release of aminomethyl coumarin (AMC) from the peptide substrate (H-Gly-Arg-AMC), whic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862KG7US Patent