Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 1' and Ligand = 'BDBM50195247'
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195247(CHEMBL3936580)copy SMILEScopy InChI
Affinity DataIC50: 0.251nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL
LigandPNGBDBM50195247(CHEMBL3936580)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z321K4PubMed