Found 17 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 4' and Ligand = 'BDBM50050525' TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:In vitro test for inhibitory activity against human dipeptidyl peptidase IV.More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.260nMpH: 2.0Assay Description:The inhibitor solution is prepared by dissolving 3-5 mg of inhibitor in pH 2 solution (0.01 N HCl), such that the concentration of the solution is eq...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Inhibition of human DPP4 expressed in HEK293 cells using Ala-Pro-p-nitroanilide hydrochloride salt as substrate preincubated for 10 mins prior to add...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMpH: 8.0Assay Description:The inhibitor solution is prepared by dissolving 3-5 mg of inhibitor in pH 2 solution (0.01 N HCl), such that the concentration of the solution is eq...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University School of Medicine
Curated by ChEMBL
Tufts University School of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMpH: 8.0Assay Description:The inhibitor solution is prepared by dissolving 3-5 mg of inhibitor in pH 2 solution (0.01 N HCl), such that the concentration of the solution is eq...More data for this Ligand-Target Pair
