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TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:AP-1 suppression activity using freshly prepared DMSO stockMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:AP-1 suppression activity using one week old DMSO stockMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:AP-1 suppression activity using one month old DMSO stockMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:AP-1 suppression activity using two months old DMSO stockMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Ability to antagonise AP-1 transcriptional activityMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1/2(Homo sapiens (Human))
DuPont Pharmaceuticals Company
Curated by ChEMBL
DuPont Pharmaceuticals Company
Curated by ChEMBL
Affinity DataIC50: 2.48E+4nMAssay Description:AP-1 suppression activity using six months old DMSO stockMore data for this Ligand-Target Pair
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