Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity mitogen-activated protein kinase kinase 1' and Ligand = 'BDBM50391803'
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Boston University

Curated by ChEMBL
LigandPNGBDBM50391803(CHEMBL2146888)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Inhibition of MEK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Boston University

Curated by ChEMBL
LigandPNGBDBM50391803(CHEMBL2146888)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Inhibition of MEK1-mediated ERK2 T202/Y204 phosphorylation using biotinylated MBP as substrate preincubated for 30 mins measured after 100 mins by cR...More data for this Ligand-Target Pair