Compile Data Set for Download or QSAR
Found 7 Enz. Inhib. hit(s) with Target = 'Dual specificity protein kinase CLK3' and Ligand = 'BDBM50347750'
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FN1B7VPubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))TBA
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 2.17E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T1553QPubMed
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK3 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2VHRPubMed
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK3 expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by scin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571D55PubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))TBA
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))TBA
LigandPNGBDBM50347750(CHEMBL1802358)copy SMILEScopy InChI
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to CLK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571D55PubMed