BindingDB PrimarySearch

Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM50346237'

Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))TBA

BDBM50346237(9-Oxy-5,12-dihydro-7H-5,9,12-triaza-dibenzo[a,e]az...)copy SMILEScopy InChI

IC50: 1.00E+4nMAssay Description:Antagonist activity at NOP receptor in Swiss mouse vas deferens by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details

Dual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Trinity College

Curated by ChEMBL

BDBM50346237(9-Oxy-5,12-dihydro-7H-5,9,12-triaza-dibenzo[a,e]az...)copy SMILEScopy InChI

IC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli assessed as assessed as incorporation of [gamma-33P]-ATP into myelin bas...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q21836T2PubMed