Found 3 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM50391956' TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT The Arctic University of Norway
Curated by ChEMBL
UiT The Arctic University of Norway
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
3D Structure (crystal)TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT The Arctic University of Norway
Curated by ChEMBL
UiT The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 329nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT The Arctic University of Norway
Curated by ChEMBL
UiT The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 329nMAssay Description:Inhibition of DYRK1A (unknown origin) using DYRKtide as substrate by ATP regenerative NADH consuming assayMore data for this Ligand-Target Pair
