Found 6 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM50530429' TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
3D Structure (crystal)TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of DYRK1A (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET ...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Inhibition of wild type full length DYRK1A (unknown origin) in human U2OS cells assessed as reduction in pSER520 autophosphorylation incubated for 5 ...More data for this Ligand-Target Pair
