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TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of DYRK1A (unknown origin) by ADP assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK1A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK1A (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET ...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Palack£ University
Curated by ChEMBL
Palack£ University
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of wild type full length DYRK1A (unknown origin) in human U2OS cells assessed as reduction in pSER520 autophosphorylation incubated for 5 ...More data for this Ligand-Target Pair
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