BindingDB PrimarySearch

Found 2 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM7266'

Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))TBA

BDBM7266(14-bromo-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)copy SMILEScopy InChI

IC50: 1.00E+4nMAssay Description:Antagonist activity at NOP receptor in Albino guinea pig ileum assessed as effect on electrically stimulated contractionsMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Trinity College

Curated by ChEMBL

BDBM7266(14-bromo-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)copy SMILEScopy InChI

IC50: 1.00E+4nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli assessed as assessed as incorporation of [gamma-33P]-ATP into myelin bas...More data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

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Details Article
BindingDB Entry DOI: 10.7270/Q21836T2PubMed